Test
Broad spectrum, irreversible inhibitor of serine proteases
Inhibits NF-κB activation
Extensive quality control produces industry leading bioactivity and lot-to-lot consistency that instills confidence in results and ensures reproducibility. Applications: Enzyme Activity
Potent PAK inhibitor; brain penetrant and orally bioavailable
Non-competitive AMPA/kainate antagonist
Potent protein kinase D (PKD) inhibitor
Synthetic thymidine analog; used for cell proliferation assays
Firefly luciferase substrate
ATP-competitive inhibitor of IGF1R
Selective P2Y6 antagonist
Potent and selective allosteric inhibitor of PRMT3
Potent and selective G9a and GLP inhibitor
Positive allosteric modulator of α4β2 nAChRs
mTOR inhibitor; antitumor
Selective Kir3.1/3.2 (GIRK1/2) channel activator